BDBM195612 GSK467

SMILES O=c1[nH]c(Oc2cnn(Cc3ccccc3)c2)nc2cnccc12

InChI Key InChIKey=ZTYRLXUTLYBVHH-UHFFFAOYSA-N

Data  20 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 195612   

TargetLysine-specific demethylase 5B(Homo sapiens (Human))TBA
LigandPNGBDBM195612(GSK467)
Affinity DataIC50:  26nMAssay Description:Inhibition of KDM5B (unknown origin) by alphascreen assayMore data for this Ligand-Target Pair
TargetLysine-specific demethylase 5B(Homo sapiens (Human))TBA
LigandPNGBDBM195612(GSK467)
Affinity DataIC50:  26nMpH: 7.5Assay Description:The demethylase AlphaScreen assay was performed in 384-well plate format using white proxiplates (PerkinElmer), and transfer of compound (100 nl) was...More data for this Ligand-Target Pair